Akwukwo hydrogromide Raw Galantamine (69353-21-5) video
Ụdị Hydrobromide Raw Galantamine (69353-21-5) Description
Ngwakọta Ugwu Galantamine Hydrobromide bụ benzazepine nke sitere na norbelladine. A na-achọta ya na GALANTHUS na ndị ọzọ AMARYLLIDACEAE. Ọ bụ onye na-emepụta cholinesterase nke ejiji iji gbanwee mmetụta muscular nke GALLAMINE TRIETHIODIDE na TUBOCURARINE ma a mụọ ya dịka ọgwụgwọ maka ọrịa ALZHEIMER na nsogbu ndị ọzọ na-ahụ maka nsogbu usoro nsogbu.
Raw Galantamine Hydrobromide ntụ ntụ bụ ụdị nnu hydrobromide nke galantamine, alkaloid dị elu nke enwetara na synthetically ma ọ bụ n'ụzọ nkịtị site na bọlbụ na okooko osisi nke Narcissus na ọtụtụ usoro ndị ọzọ nke ezinụlọ Amaryllidaceae nwere ihe omume anticholinesterase na mmezi neurocognitive. Galantamine na-asọmpi na ntụgharị na-egbochi acetylcholinesterase, si otú ahụ na-eme ka ịta ahụhụ na imeziwanye ihe nke acetylcholine (Ach). Tụkwasị na nke ahụ, galantamine bụ ligand maka ndị na-anabata acetylcholine nicotinic, nke nwere ike ime ka ntọhapụ presynaptic nke Ach ma mee ka ndị nabatara postsynaptic rụọ ọrụ. Onye ọrụ a nwere ike imeziwanye ọrụ nhụjuanya na ọrịa Alzheimer dị nro ma dị nwayọọ ma nwee ike belata mgbaàmà nke nghọta na-akwalite ị smokingụ sịga.
Akwukwo hydrogromide Raw Galantamine (69353-21-5) Smmezi
Product Name | Akwukwo hydrogromide Raw Galantamine |
Chemical Aha | Galary; Nchịkwa; Galanthamine Galanthamine Hydrobromide; Lycoremine; Nivalin Nivaline; Razadyne; Reminyl Galanthamine hydrobromide; Akwukwo hydrogromide Raw Galantamine; 1953-04-4; Reminyl; Galanthamine (hydrobromide); |
Brand Name | Enweghị data dị |
Klaasị ọgwụ ọjọọ | Alzheimer Disease Agents, cholinesterase inhibitor |
CAS Number | 69353-21-5 |
InChIKey | QORVDGQLPPAFRS-XPSHAMGMSA-N |
molekụla Fnhazi | C17H22BrNO3 |
molekụla Wasatọ | 368.271 g / mol |
Nkịtị Monoisotopic | 367.078 g / mol |
Mgbu Point | 126-127 deg C |
Na-egbuke egbuke Point | Enweghị data dị |
Ọkara Ndụ nke Ndụ | Iwepụ ọkara ndụ: 7 awa |
Agba | White siri ike |
Sume | E nwere ike ịkụnye ya na mmiri ọkụ; enweghi mmanu na mmanya, acetone, chloroform. Obere ala na benzene, ether. |
Sịkwa akwa Tigwe | -20 Celsius C |
Antinye | nhazi cholesterase; ọgwụ |
raw Hydrobromide Galantamine ntụ ntụ (69353-21-5) Nkọwa
Galantamine Hydrobromide bụ ụdị nnu hydrobromide nke galantamine, nke a na-enweta nke ọma na nke sitere na bọlbụ na okooko osisi nke Narcissus na ọtụtụ usoro ndị ọzọ nke ezinụlọ Amaryllidaceae nwere usoro anticholinesterase na mmezi neurocognitive. Galantamine na-asọmpi na ntụgharị na-egbochi acetylcholinesterase, si otú ahụ na-eme ka ịta ahụhụ na imeziwanye ihe nke acetylcholine (Ach). Tụkwasị na nke ahụ, galantamine bụ ligand maka ndị na-anabata acetylcholine nicotinic, nke nwere ike ime ka ntọhapụ presynaptic nke Ach ma mee ka ndị nabatara postsynaptic rụọ ọrụ. Onye ọrụ a nwere ike imeziwanye ọrụ nhụjuanya na ọrịa Alzheimer dị nro ma dị nwayọọ ma nwee ike belata mgbaàmà na-emetụta abstinence na-akwalite ị relaụ sịga.
Hydrobromide Galantamine ntụ ntụ (69353-21-5) Ime ihe?
Galantamine bụ phenanthrene alkaloid na onye na-agbanwe agbanwe, asọmpi acetylcholinesterase inhibitor. Enweghi mmekorita ya na ndi ozo acetylcholinesterase. Usoro usoro ihe Galantamine chọrọ na-agụnye igbochi igbochi acetylcholinesterase, nke na-egbochi hydrolysis nke acetycholine, na-eduga n'ịba ụba nke acetylcholine na cholinergic synapses. Galantamine na-ejikọkwa ihe na nicotinic acetylcholine na-anabata ma nwee ike ime ka ndị agonists rụọ ọrụ (dị ka acetylcholine) na ndị nnabata a.
uru of Hydrobromide Galantamine ntụ ntụ (69353-21-5)
- Mee ka arụ ọrụ na-arụ ọrụ mma
- Na-ebelata mmịfụ
- Ọ bụ Antioxidant
- Nwere ike igbochi ọgwụ nsị
- Nwere ike ịnagide ọrịa shuga
- Nwere ike ịnagide oke oke
- Na-egosi Dreamid Dreaming
- Nwere ike iwepụ ihe mgbaàmà nke Autism
- Nwere ike inyere aka na Schizophrenia
- Na-eme ka ọrịa ogbu na nkwonkwo gbanwee
- Nwere ike inyere gị aka ịkwụsị ise siga
- Na-egbochi Ọrịa Brain
-atụ aro Hydrobromide Galantamine ntụ ntụ (69353-21-5) Ọgwụgwọ
Kọlọsi Hydrobromide Galantamine 16 mg / ụbọchị bụ usoro ọgwụgwọ kachasị mma maka ndị ọrịa nwere AD dị arọ, dị ka nrụpụta yiri nke a na-ahụ na 24 mg / day dose. Otú ọ dị, ndị ọrịa nwere AD dị ala ga-enweta uru ndị ọzọ site na galantamine 24 mg / ụbọchị.
mmetụta of Hydrobromide Galantamine ntụ ntụ (69353-21-5)
Mmetụta ndị na-agakarị nke Galantamine Hydrobromide ntụ ntụ gụnyere mgbatị ahụ na adịghị ike, ihe omume cardio-respiratory, nsogbu akpụkpọ ahụ, na urinary incontinence. Nara nnukwu ọgwụ dị iche iche nke Galantamine na-enweghị iwuli nwayọ elu nwekwara ike ibute nrọ na nchekasị.
Na mgbakwunye na mmetụta ndị a, mmekọrịta Galantamine na ọgwụ ndị ọzọ nwere ike ịkpata nsogbu ahụ ike. A gwara ya ka ị ghara iji oge Galantamine mee ihe mgbe ị na-ewere ọgwụ ndị ọzọ a na-etinye site n'ime ụzọ imeju ahụ (usoro cytochrome nke hepatic).
Obi dị m ụtọ, ọtụtụ n'ime mmetụta ndị dị n'elu bụ ndị dị ụkọ ma eleghị anya a ga-ezere dosing.