Raw Lorcaserin hydrochloride hemihydrate powder (856681-05-5) video
Raw Lorcaserin hydrochloride hemihydrate powder (856681-05-5) Nkọwapụta
Product Name | Raw Lorcaserin hydrochloride hemihydrate uzuzu |
Chemical Aha | Lorcaserin hydrochloride, (R) -8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine hydrochloride hemihydrate; (R) -8-chloro-2,3,4,5-tetrahydro-1-methyl-1h-3-benzazepine hydrochloride hemihydrate |
Brand Name | Belviq |
Klaasị ọgwụ ọjọọ | 5-HT2C onye nkwụnye ihe nkwụnye ihe |
CAS Number | 856681-05-5 |
InChIKey | WRZCAWKMTLRWPR-VSODYHHCSA-N |
molekụla Fnhazi | C22H32Cl4N2O |
molekụla Wasatọ | 482.31 |
Nkịtị Monoisotopic | 480.1268745 |
Mgbu Point | Enweghị data dị |
Fna-agbanyeghachi Point | Enweghị data dị |
Ọkara Ndụ nke Ndụ | Lorcaserin nwere ọkara ndụ plasma nke 11 awa |
Agba | White ntụ ntụ |
Solubility | Mgbaze mmiri 0.0709 mg / mL |
nchekwa Tigwe | Enweghị data dị |
Antinye | Raw Lorcaserin hydrochloride hemihydrate ntụ ntụ eji dị ka ọgwụ mgbochi oke ibu. O nwere ọrụ dị ka onye agụụ na-agụ agụụ na agonist serotonergic. |
Raw Lorcaserin hydrochloride hemihydrate powder (856681-05-5) Nkọwapụta
Mpekota hemihydrate nke Lorcaserin hydrochloride bụ hydrate nke bụ ụdị hemihydrate nke lorcaserin hydrochloride. Eji ya mee ọgwụ. Ọ nwere ọrụ dịka onye nkoropụ agụụ na onye agonist serotoneric. O nwere ihe odide hydrochloride.
Raw Lorcaserin hydrochloride hemihydrate ntụ ntụ bụ iji mee ihe maka oke ibu nke cholesterol dị elu, ọbara mgbali elu, ma ọ bụ ụdị 2 ọrịa shuga.
FDA kwadoro Raw Lorcaserin hydrochloride hemihydrate ntụ ntụ maka ndị mmadụ buru oke ibu (nke nwere oke nkesa, ma ọ bụ BMI, nke 30 ma ọ bụ karịa) ma ọ bụ ndị buru ibu (nke nwere BMI nke 27 ma ọ bụ n'elu) ma nwee ọ dịkarịa ala otu ibu- nsogbu ahụike dịka ụdị ọrịa shuga 2, ọbara mgbali elu ma ọ bụ cholesterol dị elu.
Raw Lorcaserin hydrochloride hemihydrate ntụ ntụ na-arụ ọrụ site na ịchịkwa agụụ - kpọmkwem site n'ịkwalite ụbụrụ ụbụrụ maka serotonin, nke na-eme ka mmetụta nke satiety na afọ ojuju kpatara. Serotonin na-emetụta ọnọdụ; ọtụtụ ọgwụ ndị na-agwọ ọrịa antidepressant na-arụ ọrụ site na igbochi nlọghachi nke serotonin ma na-echekwa ụbụrụ na-ehicha na chemical. Ndị nchọpụta na Arena na-ekwu na ọgwụ ha na-eme iji chọpụta naanị ndị na-anabata serotonin na-emetụta agụụ.
Lorcaserin hydrochloride hemihydrate ntụ ntụ (856681-05-5) Usoro nke Action
A kwadoro Lorcaserin iji belata nri oriri ma kwalite satiety site na ịmepụta ndị natara 5-HT2C na pro-opiomelanocortin neurons nke dị na hypothalamus. A maghị usoro usoro nke a.
Lorcaserin na ntinye ụbọchị a na-atụ aro ya na ndị na-anata 5-HT2C na nzaghachi 5-HT2A na 5-HT2B (lee 5 Table), subtypes nke ntinye 5-HT nke ọzọ, onye natara 5-HT na saịtị 5-HT .
ngwa nke polkloride hydrochloride hemihydrate (856681-05-5)
- Onye na-enye obi ụtọ: Onye na-eme ihe iji belata agụụ.
- serotonergic agonist: Otu onye na-ahụ maka ndị na-anabata serotonin ma nwee ike ịkọ mmetụta nke serotonin site na ịme ka ọrụ ahụike dị na ndị nabatara cell. A na-eji agonists Serotonin mee ihe dị ka antidepressants, anxiolytics, na ịgwọ ọrịa ọrịa migraine.
Na-atụ aro polkloride hydrochloride hemihydrate (856681-05-5)
Ebe ọ bụ na enweghi ike ịchọta ihe ọmụma dị mkpa banyere iji Lorcaserin hydrochloride hemihydrate, ihe ndị na-esonụ bụ maka ntụle naanị:
Akwukwo nke 846589-98-8 na-abịa na mbadamba ụrọ ma na-ewere 1-2 ugboro ugboro n'ụbọchị, na-enweghị nri. A ghaghị iji mpaghara a na-eji cacarie eme ihe na usoro ihe omumu.
Ụdị a na-atụ aro maka ụbụrụ bụ 10 mg na-eji ọnụ ekwu ugboro abụọ n'ụbọchị. Enwere ike ịnabata Lorcaserin n'emeghị nri. A ghaghị ịkwụsị na ndị ọrịa bụ ndị na-emezughị iji nweta 5% nhalata ọnwụ site na izu 12 ebe ọ bụ na ndị ọrịa a agaghị enwe mmerụ ahụ dị mkpa na ọgwụgwọ na-aga n'ihu.
uru nke Fọl hemihydrate Lorcaserin hydrochloride (856681-05-5)
Ọkpụkpụ hemihydrate Lorcaserin hydrochloride bụ onye na-emepụta aghara aghara nke 5-HT2C nke a na-eche iji belata nri oriri site na usoro POMC kachasị. Lorcaserin HCL ntụ ntụ uru:
- A na-eji ntụ ntụ hemihydrate Lorcaserin hydrochloride mee ihe na nri na mmega ahụ iji na-emeso oke ibu.
- A na-ejikarị mmiri na-eme ka a na-ejikarị mmiri ozuzo na-agwọ ọrịa shuga, cholesterol dị elu, ma ọ bụ ọbara mgbali elu.
- Lorcaserin hydrochloride hemihydrate ntụ ntụ agaghị agwọ ọrịa ọ bụla (dịka ọrịa obi, ọrịa shuga, ọbara mgbali elu).
mmetụta nke polkloride hydrochloride hemihydrate (856681-05-5)
A na-eji Lorcaserin hydrochloride hemihydrate ntụ ntụ mee ihe maka ọgwụgwọ nke ịdị arọ na-adịghị ala ala na ndị okenye nwere nchịkọta anụ ahụ (BMI) nke 30 ma ọ bụ karịa (obese) dị ka mgbakwunye na nri na kalori na-ebelata. A kwadoro ya ka ndị okenye nwere BMI nke 27 ma ọ bụ karịa (buru ibu) ma nwee opekata mpe otu ọnọdụ metụtara oke dị ka ọbara mgbali elu (ọbara mgbali elu), ma ọ bụ cholesterol dị elu (dyslipidemia). Agbanyeghị, ọ nwekwara ike ịnwe ụfọdụ nsonaazụ. Dị ka n'okpuru:
Tọ bụ mmetụta kachasị emetụta ya:
- -Na-amacha,
- -Dizziness,
- -Nke ike,
- -Nausea,
- -Ndị ọnụ,
- -Constipation, na
- -Hypoglycemia (ọbara ọbara ala).
Ihe ndị ọzọ na-adịghị ahụkarị ma ọ bụ dị egwu na-emetụta ya na lorcaserin gụnyere:
- - Nsogbu valve ụkwụ,
- - Ngbanwe na anya ma ọ bụ ebe nchekwa,
- - Nsogbu uche,
- -Dress or echiche nke igbu onwe,
- -Akwado ihe ndi ozo,
- -Ka obi ghara iru gi ala,
- -Abelata ụlọnga ọbara, na
- -Anwekwu na hormone, prolactin.